Kinetics of the β2 Adrenergic receptor binding and signaling


More speed, less haste: a look at the kinetics of cAMP production in cells.

The application of kinetics to research and development for G-protein-coupled Receptor drugs has become increasingly valuable. Taking the β2-adrenergic receptor as an example, this application note provides a new integrated approach to measuring the kinetics of agonist binding and the rate of cAMP production over time.
From the data generated, an in-depth pharmacological profile of the compound tested emerges.