Download your 3 application notes on kinase inhibitor selection for kinase binding assays

3AN itk

Challenge kinase binding assays and win with HTRF technology

The 3 application notes present a new HTRF kinase binding assay that combines the usage of a fluorescent inhibitor with a tagged kinase enzyme and its corresponding anti-tag-Europium labeled detection reagent.

These 3 application notes will provide you with:

  • Validation data for the 3 fluorescent tracers  Dasatinib-red, Staurosporine-red and Sunitinib-red
  • Guidance for the determination of inhibitor constants: Kd and Ki
  • Pharmacological characterization of known inhibitors and correlation with literature data
  • Relevant case studies to help you revolutionize your assays